Tocris Bioscience
Saxagliptin hydrochloride
6507
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Saxagliptin is correlated to increased hospitalization for heart failure. We treated cardiomyocytes and followed phosphorylation of CaMKII. Saxagliptin treatment inhibited CaMKII phosphorylation in a concentration dependent manner.
Cell culture
Cardiomyocytes
N/A
Saxagliptin reduced pCaMKII expression in cardiomyocytes. This resulted in impaired calcium homeostasis.
Worked as expected
Saxagliptin impairs CaMKII activity and calcium homeostasis in cardiomyocytes.