Description
A positive allosteric modulator of 5-HT2A and 5-HT2C receptors; selective for these receptors over a panel of 21 receptors and transporters at 10 µM; enhances 5-HT-induced calcium release in CHO cells expressing recombinant human 5-HT2A or 5-HT2C at 1 nM; reduces spontaneous locomotor activity in rats at 30 mg/kg