Description
EA4, a derivative of quinone, is an inhibitor for both rPLA and cPLA. EA4 can inhibit rPLA 2 with a K i value of 130 µM. EA4 can be used for the research of hemostasis, thrombosis, and erythropoiesisIn VitroEA4 (9 µM, 24 µM) inhibits both rPLA 2 and cPLA 2. EA4 can inhibit rPLA 2 with a K i value of 130 µM. EA4 (50 µM) significantly inhibits A23187-induced AA release from both human and bovine RBCs in a time-dependent manner. MCE has not independently confirmed the accuracy of these methods. They are for reference only.Form:SolidIC50& Target:Ki: 130 µM (rPLA 2 )