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Protein Biochemistry
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limertinib
limertinib from MedChemExpress
Be the first to write a review!
Citations:
(3)
Supplier Page
Supplier Page from
MedChemExpress for
limertinib
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Description
limertinib (ASK120067) is a potent and orally active inhibitor of
EGFR
T790M
(
IC
50
:0.3 nM) with selectivity over EGFR
WT
(IC
50
:6.0 nM). limertinib is a third-generation EGFR-TKI for the research of non-small cell lung cancer (NSCLC)
Product Specs
Company Info
Citations
Reviews
Product Specs
Item
limertinib
Company
MedChemExpress
Price
$204.00
Supplier Page
View Company Product Page
Catalog Number
HY-138751
Quantity
10 mM * 1 mL
Applications
Bioactivity, Structure and function analysis, ELISA, SDS-PAGE, Western blotting
Purity
99.12%
Type
Chemical
Molecular Weight
546.06
Formula
C₂₉H₃₂ClN₇O₂
Research Area
Cancer
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MedChemExpress
1 Deer Park Drive, Suite F
MONMOUTH JUNCTION
,
NJ
08852
United States
Phone
: US Tel: 609-228-6898
US Fax: 609-228-5909
EU Tel: +4686500910
Email: sales@medchemexpress.com
eu.sales@MedChemExpress.com
Company Profile
Website:
medchemexpress.com
Citations (3)
(1)
High-throughput screening identifies NT-1 that synergizes with MRTX1133 against acquired resistant KRASG12D colorectal cancer
npj Precision Oncology
April 8, 2026
Natalie Thielen, Ning Wei, Emiko Nagai, Michele Houston, Leonard H. Augenlicht, Alice E. Shin, Joel T. Gabre, Anil K. Rustgi, Grace Ha, Lindsay M. LaFave,
et al.
NT-1 (
Mutant EGFR Inhibitor
,
HY-13984
),
ASN007
(
HY-136579
),
p38α inhibitor 2
(
HY-131335
),
Limertinib
(
HY-138751
),
CDK8-IN-4
(
HY-111465
),
CDK12-IN-E9
(
HY-117203A
),
Osimertinib
(
HY-15772
), Afatinib (HY-10261), Gefitinib
(2)
Profiling and Optimizing Targeted Covalent Inhibitors through EGFR-Guided Studies
Journal of Medicinal Chemistry
August 28, 2025
Tahereh Damghani, Surbhi P. Chitnis, Omobolanle A. Abidakun, Kishan B. Patel, Kaly S. Lin, Emily A. Ouellette, Abigail M. Lantry, David E. Heppner
lazertinib (Selleckchem S8724), 8 oritinib (
MedChemExpress
HY-139920
), 9 limertinib (
MedChemExpress
HY-138751
), 10 canertinib (
MedChemExpress
HY-10367
), 11 afatinib (Thermo Fisher Sci 465642500), 12 BDTX-1535 (Selleckchem
(3)
Discovery of a novel third-generation EGFR inhibitor and identification of a potential combination strategy to overcome resistance
Molecular cancer
May 13, 2020
Zhang T, Qu R, Chan S, Lai M, Tong L, Feng F, Chen H, Song T, Song P, Bai G,
et al
.
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limertinib from MedChemExpress
Supplier Page
View Company Product Page
$204.00
Product Specs
Company Info
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