CMPD101 from BOC Sciences

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Supplier Page from
BOC Sciences for
CMPD101

Description

CMPD101 is a selective GRK2/3 inhibitor with IC50 value is 54 nM for GRK3 and 32 nM for GRK2. It shows selectivity for GRK2/3 over GRK1/5. It can also reduce DAMGO-induced desensitization and internalization of µ-opioid receptors