AMG 9810 from Tocris Bioscience, a Bio-Techne Brand

Product Specs
ItemAMG 9810
CompanyTocris Bioscience, a Bio-Techne Brand
Price $228.00Supplier Page View Company Product Page
Catalog Number2316/10
Quantity10 mg (also 50 mg)
Purity98%
Molecular Weight337.42
Molecule Name(2E)-N-(2,3-Dihydro-1,4-benzodioxin-6-yl)-3-[4-(1,1-dimethylethyl)phenyl]-2-propenamide
FormulaC21H23NO3
StorageStore at +4°C

Specifications/Features

Sizes Available: 10 mg (also 50 mg)

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Tocris Bioscience, a Bio-Techne Brand

614 McKinley Place N.E.

Minneapolis, Minnesota 55413

United States

Phone: 1 (800) 343-7475
1 (612) 379-2956
Fax: 1 (612) 656-4400

Company Profile

Website: http://www.tocris.com

(1) Epigenetic Upregulation of Carotid Body Angiotensin Signaling Increases Blood PressureHypertensionDecember 5, 2024Fengli Zhu, Zhuqing Wang, Kayla Davis, Hayden McSwiggin, Jekaterina Zyuzin, Jie Liu, Wei Yan, Virender K. Rehan, Nicholas JendzjowskyCat. No. 3798, 3 µM), nicotine+Ang II+losartan, Ang II+AMG9810 (TRPV1 antagonist; Tocris, Cat. No. 2316, 10 µM), nicotine+Ang II+AMG9810, or nicotine+Ang II+losartan+AMG9810. Cells were then treated with Calcium

(2) Cannabinoid combination targets NOTCH1-mutated T-cell acute lymphoblastic leukemia through the integrated stress response pathwayElifeSeptember 11, 2024Elazar Besser, Anat Gelfand, Shiri Procaccia, Paula Berman, David MeiriIsrael). The antagonists CID 16020046 (#4959/5), AM630 (#1120/10), SR-144,528 (#5039/10), and AMG9810 (#2316/10) were purchased from Tocris Bioscience (Bristol, UK). BIM-46187 (#5332990001) and ISRIB (#SML0843) were

(3) Cannabinoid combination targets NOTCH1-mutated T-cell acute lymphoblastic leukemia through the integrated stress response pathwayeLifeSeptember 11, 2024Elazar Besser, Anat Gelfand, Shiri Procaccia, Paula Berman, David MeiriIsrael). The antagonists CID 16020046 (#4959/5), AM630 (#1120/10), SR-144,528 (#5039/10), and AMG9810 (#2316/10) were purchased from Tocris Bioscience (Bristol, UK). BIM-46187 (#5332990001) and ISRIB (#SML0843) were

(4) The Effect of Cannabis Plant Extracts on Head and Neck Squamous Cell Carcinoma and the Quest for Cannabis-Based Personalized TherapyCancersJanuary 13, 2023Blal K, Besser E, Procaccia S, Schwob O, Lerenthal Y, Abu Tair J, Meiri D, Benny O.lyophilized to dryness and analyzed by UHPLC/UV and ESI-LC/MS. 2.4. Reagents Am630 (#1120/10), AMG9810 (#2316/10), and SET2 (6990/10) were purchased from Tocris Bioscience (Bristol, UK). BIM-46187 (#5332990001) and

(5) Combination of a Rapidly Penetrating Agonist and a Slowly Penetrating Antagonist Affords Agonist Action of Limited Duration at the Cellular LevelBiomolecules & therapeuticsSeptember 1, 2019Pearce LV, Ann J, Blumberg PM, Lee J.

(6) fMRI indicates cortical activation through TRPV1 modulation during acute gouty attacksScientific reportsAugust 26, 2019Chen CC, Chang C, Hsu YH, Peng YJ, Lee HS, Huang GS.

(7) Lionfish venom elicits pain predominantly through the activation of nonpeptidergic nociceptorsPainNovember 1, 2018Mouchbahani-Constance S, Lesperance LS, Petitjean H, Davidova A, Macpherson A, Prescott SA, Sharif-Naeini R.

(8) Activation of temperature-sensitive TRPV1-like receptors in ARC POMC neurons reduces food intakePLoS biologyApril 1, 2018Jeong JH, Lee DK, Liu SM, Chua SC Jr, Schwartz GJ, Jo YH.

(9) Epiregulin and EGFR interactions are involved in pain processingThe Journal of clinical investigationSeptember 1, 2017Martin LJ, Smith SB, Khoutorsky A, Magnussen CA, Samoshkin A, Sorge RE, Cho C, Yosefpour N, Sivaselvachandran S, Tohyama S, et al.

(10) The medullary dorsal reticular nucleus as a relay for descending pronociception induced by the mGluR5 in the rat infralimbic cortexNeuroscienceMay 4, 2017David-Pereira A, Sagalajev B, Wei H, Almeida A, Pertovaara A, Pinto-Ribeiro F.

(11) IL-33/ST2 signaling excites sensory neurons and mediates itch response in a mouse model of poison ivy contact allergyProceedings of the National Academy of Sciences of the United States of AmericaNovember 22, 2016Liu B, Tai Y, Achanta S, Kaelberer MM, Caceres AI, Shao X, Fang J, Jordt SE.

(12) The Complement System Component C5a Produces Thermal Hyperalgesia via Macrophage-to-Nociceptor Signaling That Requires NGF and TRPV1The Journal of neuroscience : the official journal of the Society for NeuroscienceMay 4, 2016Shutov LP, Warwick CA, Shi X, Gnanasekaran A, Shepherd AJ, Mohapatra DP, Woodruff TM, Clark JD, Usachev YM.

(13) The Cancer Chemotherapeutic Paclitaxel Increases Human and Rodent Sensory Neuron Responses to TRPV1 by Activation of TLR4The Journal of neuroscience : the official journal of the Society for NeuroscienceSeptember 30, 2015Li Y, Adamek P, Zhang H, Tatsui CE, Rhines LD, Mrozkova P, Li Q, Kosturakis AK, Cassidy RM, Harrison DS, et al.

(14) Mother root of Aconitum carmichaelii Debeaux exerts antinociceptive effect in Complet Freund's Adjuvant-induced mice: roles of dynorpin/kappa-opioid system and transient receptor potential vanilloid type-1 ion channelJournal of translational medicineAugust 30, 2015Wang C, Sun D, Liu C, Zhu C, Jing X, Chen S, Liu C, Zhi K, Xu T, Wang H, et al.

(15) Endocannabinoids Mediate Muscarinic Acetylcholine Receptor-Dependent Long-Term Depression in the Adult Medial Prefrontal CortexFrontiers in cellular neuroscienceJanuary 1, 2015Martin HG, Bernabeu A, Lassalle O, Bouille C, Beurrier C, Pelissier-Alicot AL, Manzoni OJ.

(16) The endocannabinoid/endovanilloid N-arachidonoyl dopamine (NADA) and synthetic cannabinoid WIN55,212-2 abate the inflammatory activation of human endothelial cellsThe Journal of biological chemistryMay 9, 2014Wilhelmsen K, Khakpour S, Tran A, Sheehan K, Schumacher M, Xu F, Hellman J.

(17) P2X₃ and TRPV1 functionally interact and mediate sensitization of trigeminal sensory neuronsNeuroscienceMarch 1, 2013Saloman JL, Chung MK, Ro JY.

(18) Plant derived aporphinic alkaloid S-(+)-dicentrine induces antinociceptive effect in both acute and chronic inflammatory pain models: evidence for a role of TRPA1 channelsPloS oneJanuary 1, 2013Montrucchio DP, Córdova MM, Santos AR.

(19) 5,6-EET is released upon neuronal activity and induces mechanical pain hypersensitivity via TRPA1 on central afferent terminalsThe Journal of neuroscience : the official journal of the Society for NeuroscienceMay 2, 2012Sisignano M, Park CK, Angioni C, Zhang DD, von Hehn C, Cobos EJ, Ghasemlou N, Xu ZZ, Kumaran V, Lu R, et al.

(20) Endocannabinoid System and TRPV1 Receptors in the Dorsal Hippocampus of the Rats Modulate Anxiety-like BehaviorsIranian journal of basic medical sciencesMay 1, 2012Hakimizadeh E, Oryan S, Hajizadeh Moghaddam A, Shamsizadeh A, Roohbakhsh A.

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AMG 9810

AMG 9810 from Tocris Bioscience, a Bio-Techne Brand

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Specifications/Features

Tocris Bioscience, a Bio-Techne Brand

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AMG 9810 from Tocris Bioscience, a Bio-Techne Brand

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