CMPD101 from Tocris Bioscience, a Bio-Techne Brand | Biocompare.com

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CMPD101

Potent and selective GRK2/3 inhibitor

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Tocris Bioscience, a Bio-Techne Brand for
CMPD101

Description

Potent and selective GRK2/3 inhibitor

Product Specs
ItemCMPD101
CompanyTocris Bioscience, a Bio-Techne Brand
Price $225.00Supplier Page View Company Product Page
Catalog Number5642/10
Quantity10 mg
Purity98%
Molecular Weight466.46
Molecule Name3-[[[4-Methyl-5-(4-pyridinyl)-4H-1,2,4-triazol-3-yl]methyl]amino]-N-[[2-(trifluoromethyl)phenyl]methyl]benzamide
FormulaC24H21F3N6O
StorageStore at -20°C

Specifications/Features

Sizes Available: 10 mg

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Tocris Bioscience, a Bio-Techne Brand

614 McKinley Place N.E.

Minneapolis, Minnesota 55413

United States

Phone: 1 (800) 343-7475
1 (612) 379-2956
Fax: 1 (612) 656-4400

Company Profile

Website: http://www.tocris.com

(1) Subcellular location defines GPCR signal transductionScience advancesApril 21, 2023Radoux-Mergault A, Oberhauser L, Aureli S, Gervasio FL, Stoeber M.

(2) Mechanical and chemical activation of GPR68 probed with a genetically encoded fluorescent reporterJournal of cell scienceAugust 15, 2021Ozkan AD, Gettas T, Sogata A, Phaychanpheng W, Zhou M, Lacroix JJ.

(3) Biological characterization of ligands targeting the human CC chemokine receptor 8 (CCR8) reveals the biased signaling properties of small molecule agonistsBiochemical pharmacologyJune 1, 2021Liu L, Doijen J, D'huys T, Verhaegen Y, Dehaen W, De Jonghe S, Schols D, Van Loy T.

(4) Mechanisms of differential desensitization of metabotropic glutamate receptorsCell reportsApril 27, 2021Abreu N, Acosta-Ruiz A, Xiang G, Levitz J.

(5) Mutations in GRK2 cause Jeune syndrome by impairing Hedgehog and canonical Wnt signalingEMBO molecular medicineNovember 6, 2020Bosakova M, Abraham SP, Nita A, Hruba E, Buchtova M, Taylor SP, Duran I, Martin J, Svozilova K, Barta T, et al.

(6) A Discrete Presynaptic Vesicle Cycle for Neuromodulator ReceptorsNeuronFebruary 19, 2020Jullié D, Stoeber M, Sibarita JB, Zieger HL, Bartol TM, Arttamangkul S, Sejnowski TJ, Hosy E, von Zastrow M.

(7) Conformational signatures in β-arrestin2 reveal natural biased agonism at a G-protein-coupled receptorCommunications biologyJanuary 1, 2018Reyes-Alcaraz A, Lee YN, Yun S, Hwang JI, Seong JY.

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