Description
InformationBatefenterol (GSK961081, TD-5959) is both amuscarinic receptorantagonist and aβ2-adrenoceptoragonist with Ki of 1.4 nM, 1.3 nM and 3.7 nM for hM2, hM3 muscarinic receptors and hβ2-adrenoceptor, respectively.TargetshM3 muscarinic receptor (Cell-free assay); hM2 muscarinic receptor (Cell-free assay); hβ2-adrenoceptor (Cell-free assay) 1.3 nM(Ki); 1.4 nM(Ki); 3.7 nM(Ki)