Description
A Bax inhibitor; binds to Bax in a cell-free assay (Kd = 15 µM); inhibits tBID-induced Bax-mediated membrane permeabilization in a liposomal release assay (IC50 = 3.3 µM); inhibits TNF-α- and cycloheximide-induced apoptosis in MEFs (IC50 = 1.8 µM); inhibits BTSA1-induced cell death in OCI-AML-3 cells