Welcome Guest
Sign In
Register
Products
Popular Categories
Antibody Search
ELISA Kit Search
Biomolecules
Flow Cytometers
Thermal Cyclers
Microscopes
Transfection Reagents
Featured Products
New Products
Research Areas
ELISA
Western Blot
3D Cell Culture
Digital PCR
Quantitative PCR
Cell and Gene Therapy
In Vivo Models
Resources
eBooks
Bench Tips
Tech Insights
Editorial Articles
News
Product Reviews
Future Lab
White Papers
Infographics
Events
Promotions
Multimedia
Biocompare Webinars
Technologies Transforming Precision Medicine
Immunotherapy
Reproducibility
Transformative Technologies
Podcasts
Bench Tip Videos
All Videos and Webinars
Life Science Webinars
Write a Review
Antibodies
Kits/Reagents
Equipment
Services
Register
Sign In
Biocompare
Products
Protein Biochemistry
Chemicals and Reagents
GK921
GK921 from MedChemExpress
Be the first to write a review!
Citations:
(6)
Supplier Page
Supplier Page from
MedChemExpress for
GK921
Get Pricing
Description
GK921 is a transglutaminase 2 (
TGase
) inhibitor with an
IC
50
of 7.71 µM for human recombinant TGase 2
Product Specs
Company Info
Citations
Reviews
Product Specs
Item
GK921
Company
MedChemExpress
Price
$104.00
Supplier Page
View Company Product Page
Catalog Number
HY-12337
Quantity
10 mM * 1 mL
Applications
Bioactivity, Structure and function analysis, ELISA, SDS-PAGE, Western blotting
Purity
99.91%
Type
Chemical
Molecular Weight
344.41
Formula
C₂₁H₂₀N₄O
Research Area
Cancer
Add to Compare List
MedChemExpress
1 Deer Park Drive, Suite F
MONMOUTH JUNCTION
,
NJ
08852
United States
Phone
: US Tel: 609-228-6898
US Fax: 609-228-5909
EU Tel: +4686500910
Email: sales@medchemexpress.com
eu.sales@MedChemExpress.com
Company Profile
Website:
medchemexpress.com
Citations (6)
(1)
Interaction of NDRG1 and TGM2 modulates DNA replication and repair
Mol Cancer Res
March 31, 2026
Hanna M. Doh, Nina Kozlova, Kayla A. Cruz, Taru Muranen
(616467, Sigma-Aldrich) was reconstituted in DMSO and used at a final concentration of 50 μM.
GK921
(
HY-12337
,
MedChemExpress
) was reconstituted in DMSO and used at a final concentration
of 1
μM. SYBR™ Gold Nucleic
(2)
Interaction of NDRG1 and TGM2 modulates DNA replication and repair
Molecular Cancer Research
March 31, 2026
Hanna M. Doh, Nina Kozlova, Kayla A. Cruz, Taru Muranen
(616467, Sigma-Aldrich) was reconstituted in DMSO and used at a final concentration of 50 μM.
GK921
(
HY-12337
,
MedChemExpress
) was reconstituted in DMSO and used at a final concentration
of 1
μM. SYBR™ Gold Nucleic
(3)
Serotonin promotes lip sensory recovery after inferior alveolar nerve transection via histone serotonylation
Journal of Dental Sciences
October 1, 2025
Suning Mao, Gaowei Zhang, Pingchuan Ma, Zhongkai Ma, Chunjie Li, Li Ye
Serotonin hydrochloride
(
HY–B1473
,
MedChemExpress
, Middlesex, NJ, USA) or 50 μM transglutaminase 2
inhibitor
GK921
(
HY-12337
,
MedChemExpress
).
Cell culture
The trigeminal
ganglion
tissues of postnatal
mice
were separated from
(4)
Fatostatin delayed lip sensory recovery after inferior alveolar nerve transection by inhibiting sterol regulatory element-binding protein 1
Journal of Dental Sciences
July 1, 2025
Suning Mao, Zhongkai Ma, Gaowei Zhang, Pingchuan Ma, Chunjie Li, Li Ye
inferior alveolar nerve transection model was established as we previously described.2 100 μM fatostatin (
HY-12337
,
MedChemExpress
, Monmouth Junction, NJ, USA) was administered to trigeminal ganglia through the infraorbital
(5)
Transglutaminase 2 nuclear localization enhances glioblastoma radiation resistance
Discov Oncol
May 30, 2025
Cuiping Sun, Zhiyong Du, Wenhui Yang, Qing Wang
Proteintech, Rosemont, IL, USA). The
inhibitors
Cystamine dihydrochloride
(Cys-D) (
HY-W020050
) and
GK921
(
HY-12337
) were obtained from
MCE
(Monmouth Junction, NJ, USA). Patient samples
Glioma
tissue
microarray
was
(6)
Transglutaminase 2 inhibitor abrogates renal cell carcinoma in xenograft models
Journal of cancer research and clinical oncology
May 1, 2014
Ku BM, Kim SJ, Kim N, Hong D, Choi YB, Lee SH, Gong YD, Kim SY.
<<
<
>
>>
Reviews
Be the First to Write a Review!
GK921 from MedChemExpress
Supplier Page
View Company Product Page
$104.00
Product Specs
Company Info
Citations
Reviews
Back To Top