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Galeterone
Galeterone from MedChemExpress
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Citations:
(5)
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Galeterone
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Description
Galeterone (TOK-001) is a multifunctional antiandrogen and
CYP17
inhibitor (
IC
50
=47 nM) in castration resistant prostate cancer (CRPC)
Product Specs
Company Info
Citations
Reviews
Product Specs
Item
Galeterone
Company
MedChemExpress
Price
$73.00
Supplier Page
View Company Product Page
Catalog Number
HY-70006
Quantity
10 mM * 1 mL
Applications
Bioactivity, Structure and function analysis, ELISA, SDS-PAGE, Western blotting
Purity
99.87%
Type
Chemical
Molecular Weight
388.55
Molecule Name
Galeterone
Formula
C26H32N2O
Research Area
Cancer
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MedChemExpress
1 Deer Park Drive, Suite F
MONMOUTH JUNCTION
,
NJ
08852
United States
Phone
: US Tel: 609-228-6898
US Fax: 609-228-5909
EU Tel: +4686500910
Email: sales@medchemexpress.com
eu.sales@MedChemExpress.com
Company Profile
Website:
medchemexpress.com
Citations (5)
(1)
Salinization Dramatically Enhance the Anti-Prostate Cancer Efficacies of AR/AR-V7 and Mnk1/2 Molecular Glue Degraders, Galeterone and VNPP433-3β Which Outperform Docetaxel and Enzalutamide in CRPC CWR22Rv1 Xenograft Mouse Model
Bioorganic chemistry
October 1, 2023
Thankan RS, Thomas E, Purushottamachar P, Weber DJ, Njar VCO.
(2)
Direct regulation of androgen receptor activity by potent CYP17 inhibitors in prostate cancer cells
The Journal of biological chemistry
February 3, 2012
Soifer HS, Souleimanian N, Wu S, Voskresenskiy AM, Collak FK, Cinar B, Stein CA.
(3)
Structures of cytochrome P450 17A1 with prostate cancer drugs abiraterone and TOK-001
Nature
January 22, 2012
DeVore NM, Scott EE.
(4)
Synthesis and biological evaluations of putative metabolically stable analogs of VN/124-1 (TOK-001): head to head anti-tumor efficacy evaluation of VN/124-1 (TOK-001) and abiraterone in LAPC-4 human prostate cancer xenograft model
Steroids
November 1, 2011
Bruno RD, Vasaitis TS, Gediya LK, Purushottamachar P, Godbole AM, Ates-Alagoz Z, Brodie AM, Njar VC.
(5)
Treatment of renal-cell cancer by transplantation of allogeneic stem cells
The New England journal of medicine
January 11, 2001
Spitzer TR, Sykes M.
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Galeterone from MedChemExpress
Supplier Page
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$73.00
Product Specs
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