Description
BAZ2-ICR is a potent, selective and cell-active inhibitor of BAZ2A (Kd=109nM; IC50=130nM) and BAZ2B (Kd=170nM; IC50=180nM) bromodomains; demonstrates 15-fold selectivity for binding BAZ2A/B over CECR2 and >100-fold selectivity over all other bromodomains