Bitopertin R enantiomer from MyBioSource.com

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Bitopertin R enantiomer

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Description

A potent and selective GlyT1 inhibitor with EC50 of 54nM; no activity for GlyT2, hERG, CYP450 enzymes above 10uM; the R enantiomer of RG-1678. Schizophrenia Phase 3 Clinical