Adenosine Kinase Inhibitor (hydrate) from Cayman Chemical

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Adenosine Kinase Inhibitor (hydrate)

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Description

A non-nucleoside pyridopyrimidine compound that selectively blocks the action of adenosine kinase in an adenosine-competitive manner (IC50 = 1.7 nM in cell-free assays); suppresses nociception in various rodent pain models