Description
An NMDA receptor agonist; binds to NMDA receptors (Ki = 0.052 µM); is selective for NMDA over kainate and AMPA receptors in radioligand binding assays (Kis = >300 µM for both); induces inward currents in Xenopus oocytes expressing rat NMDA receptors (EC50 = 1.26 µM); induces contralateral turning in rats at 30 and 70 nmol/animal