Description
A PCKζ inhibitor; 8,000-, 20,671-, 711-, 918-, 1,895-, 12,424-, 10-, and 1,218-fold selective for PKCζ over PKCα, PKCβII, PKCγ, PKCδ, PKCε, PKCη, PKCι, and PKCθ, respectively; inhibits 27 additional kinases in a panel of 37 kinases at 10 µM