Description
Idazoxan hydrochloride is an alpha2-AR adrenoceptor antagonist and potential I2 imidazoline receptor agonist. Also displays I1 imidazoline receptor antagonist activity. (pKi values are 5.90, 7.22, 8.01, 7.43, and 7.7 for I1, I2, alpha 2A, alpha2B, and alpha 2C receptors respectively)