Tranylcypromine (2-PCPA) 27305 from BPS Bioscience, Inc.

Description

Tranylcypromine (2-PCPA) is an irreversible inhibitor of LSD1 histone demethylase and monoamine oxidases (MAO). The inhibitor targets monoamine oxidases A and B and has been used as a chemical scaffold to design new demethylase inhibitors. Tranylcypromine has been shown to increase Histone H3 lysine 4 (H3K4) methylation in P19 embryonal carcinoma cell

Product Specs
ItemTranylcypromine (2-PCPA)
CompanyBPS Bioscience, Inc.
Price $215.00Supplier Page View Company Product Page
Catalog Number27305
Size1 g
ActivityTranylcypromine inhibits LSD1 with an IC50 value of 20.7 µM and a Ki value of 242.7 µM. It also irreversibly inhibits MAO A and MAO B with IC50 values of 2.3 and 0.95 µM and Ki values of 101.9 and 16 µM, respectively
Purity≥98% by HPLC
Molecular Weight364.5 kDa
FormulaC₁₈H₂₂N₂ • H₂SO₄
TypeInhibitor
FormatWhite to off-white solid