GSK256066 27751-2 from BPS Bioscience, Inc.

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GSK256066

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BPS Bioscience, Inc. for
GSK256066

Description

GSK256066 is a selective PDE4 inhibitor with an exceptionally high-affinity and selective inhibitor of phosphodiesterase 4 vs. other PDE isoforms. Often used clinically by inhalation in chronic obstructive pulmonary disease and asthma

Product Specs
ItemGSK256066
CompanyBPS Bioscience, Inc.
Price $800.00Supplier Page View Company Product Page
Catalog Number27751-2
Size50 mg
ActivityIC50 =3.2 pM for PDE4B, with >380,000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7. GSK256066 inhibits PDE4 isoforms A-D with equal affinity
Molecular Weight518.6 Da
FormulaC₂₇H₂₆N₄O₅S
TypePDE Inhibitor
TargetPDE4