GSK 2837808A from Tocris Bioscience, a Bio-Techne Brand

Product Specs
ItemGSK 2837808A
CompanyTocris Bioscience, a Bio-Techne Brand
Price Pricing Info Supplier Page View Company Product Page
Catalog Number5189/10
Quantity10 mg
Purity0.98
Molecular Weight649.62
Molecule Name3-[[3-[(Cyclopropylamino)sulfonyl]-7-(2,4-dimethoxy-5-pyrimidinyl)-4-quinolinyl]amino]-5-(3,5-difluorophenoxy)benzoic acid
FormulaC₃₁H₂₅F₂N₅O₇S
Brand/TrademarkTocris, a Bio-Techne Brand
StorageStore at -20°C

614 McKinley Place N.E.

Minneapolis, Minnesota 55413

United States

Phone: 1 (800) 343-7475
1 (612) 379-2956
Fax: 1 (612) 656-4400

(1) Mitochondrial pyruvate metabolism regulates the activation of quiescent adult neural stem cellsScience advancesMarch 1, 2023Petrelli F, Scandella V, Montessuit S, Zamboni N, Martinou JC, Knobloch M.

(2) Lactate exposure shapes the metabolic and transcriptomic profile of CD8+ T cellsFrontiers in immunologyJanuary 1, 2023Barbieri L, Veliça P, Gameiro PA, Cunha PP, Foskolou IP, Rullman E, Bargiela D, Johnson RS, Rundqvist H.

(4) Tumor-Derived Lactic Acid Modulates Activation and Metabolic Status of Draining Lymph Node StromaCancer immunology researchApril 1, 2022Riedel A, Helal M, Pedro L, Swietlik JJ, Shorthouse D, Schmitz W, Haas L, Young T, da Costa ASH, Davidson S, et al.

(5) Fructose reprogrammes glutamine-dependent oxidative metabolism to support LPS-induced inflammationNature communicationsFebruary 22, 2021Jones N, Blagih J, Zani F, Rees A, Hill DG, Jenkins BJ, Bull CJ, Moreira D, Bantan AIM, Cronin JG, et al.

(6) The distinct roles of calcium in rapid control of neuronal glycolysis and the tricarboxylic acid cycleeLifeFebruary 8, 2021Díaz-García CM, Meyer DJ, Nathwani N, Rahman M, Martínez-François JR, Yellen G.

(7) Metabolic reprogramming of osteoclasts represents a therapeutic target during the treatment of osteoporosisScientific reportsDecember 3, 2020Taubmann J, Krishnacoumar B, Böhm C, Faas M, Müller DIH, Adam S, Stoll C, Böttcher M, Mougiakakos D, Sonnewald U, et al.

(8) Lactate production is a prioritized feature of adipocyte metabolismThe Journal of biological chemistryJanuary 3, 2020Krycer JR, Quek LE, Francis D, Fazakerley DJ, Elkington SD, Diaz-Vegas A, Cooke KC, Weiss FC, Duan X, Kurdyukov S, et al.

(9) Increased Tumor Glycolysis Characterizes Immune Resistance to Adoptive T Cell TherapyCell metabolismMay 1, 2018Cascone T, McKenzie JA, Mbofung RM, Punt S, Wang Z, Xu C, Williams LJ, Wang Z, Bristow CA, Carugo A, et al.

(10) Cancer cell metabolic plasticity allows resistance to NAMPT inhibition but invariably induces dependence on LDHACancer & metabolismJanuary 1, 2018Thongon N, Zucal C, D'Agostino VG, Tebaldi T, Ravera S, Zamporlini F, Piacente F, Moschoi R, Raffaelli N, Quattrone A, et al.

(12) Neuronal Stimulation Triggers Neuronal Glycolysis and Not Lactate UptakeCell metabolismAugust 1, 2017Díaz-García CM, Mongeon R, Lahmann C, Koveal D, Zucker H, Yellen G.

(16) Breaking Cryo-EM Resolution Barriers to Facilitate Drug DiscoveryCellJune 16, 2016Merk A, Bartesaghi A, Banerjee S, Falconieri V, Rao P, Davis MI, Pragani R, Boxer MB, Earl LA, Milne JLS, et al.

GSK 2837808A