AM-251 from Enzo Life Sciences, Inc.

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Enzo Life Sciences, Inc. for
AM-251

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Description

Cannabinoid CB 1 receptor antagonist (K i =7.5 nM). Displays a high level of selectivity (306-fold) for CB 1 over CB 2 receptors. Structurally related to the cannabinoid receptor (CB) antagonist SR 141716A